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廖志新,2001年6月博士毕业于兰州大学化学化工学院天然有机化学专业,师从陈耀祖院士;2001年7月-2003年10月在中国科学院上海药物研究所天然药化研究室作博士后研究(导师,岳建民院士,期间至瑞士Novartis Pharm. AG访问进修);2003年12月-2005年12月在复旦大学药学院工作;2006年1月至今在东南大学化学化工学院工作。先后主持、参加多项国家自然科学基金、中科院重大项目及省部级科研项目的研究工作,1998年入选中央组织部、中国科学院“西部之光”人才培养计划项目。迄今发表研究论文百余篇,申请发明专利十余项,2004年作为完成人“中国龙胆科植物研究”研究成果获省级“科技进步”一等奖。主要从事天然药物的活性成分、质量、工艺研究及中药新药、药物中间体开发工作。
1.青藏高原龙胆科植物抗肝胆疾病新药源研究,中国科学院、中央组织部“西部之光”人才培养项目(主持)
2.荧光仿生膜技术研究中药活性的细胞膜通透性,国家自然科学基金项目(主要参加)
3.三种藏药植物中的VEGF抑制活性先导化合物的发现,国家自然科学基金项目(主持)
4.桂花果实抗肿瘤活性成分的发现,教育部广西师范大学药用资源化学与药物分子工程重点实验室项目(主持)
5.植提全氨基酸枸杞叶面肥产业化及关键技术研究,青海省二〇一七年重点研发与转化计划项目(主持)
6.细胞核增殖抗原(PCNA)调节浒苔快速增殖的分子机制研究,国家自然科学基金项目,(主要参加)
7.腰果高效加工及副产物综合利用关键技术研究,国家重点研发计划(子课题负责人)
1. Lei Chen, Mei Su, Qiu Jin, Wei Wang, Chun-Gu Wang, Israa Assani, Mu-Xuan Wang, Shi-Feng Zhao, Shen-Min Lv, Jia-Wei Wang, Bo Sun, Yan Li, Zhi-Xin Liao,Discovery of Chromane-6-Sulfonamide Derivative as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor t Inverse Agonist,Journal of Medicinal Chemistry,(2021),64,16106-16131
2. Yan Li, Israa Assani, Jia-Wei Wang, Chun-Gu Wang, Bo Sun, Ling-Fei Liu, Mu-Xuan Wang,Zhi Chen, and Zhi-Xin Liao,Extraction, Purification, Characterization, and Bioactive Properties of Polysaccharides from Sphallerocarpus gracilis,Starch-Stärke (2021), DOI10.1002/star.202100082
3. Ling-Fei Liu, Israa Assani, Chun-Gu Wang, Lei Chen, Bo Sun, Yan Li, Zhi Chen,and Zhi-Xin Liao,A New Triterpene, Chemical Composition, Antioxidant and In Vitro Cytotoxic Activities of Hedyotis uncinella,ChemistrySelect (2021),6, 4207 – 4211
4. Bo Sun, Israa Assani, Chun-Gu Wang, Mu-Xuan Wang, Ling-Fei Liu, Yan Li, Ge,Yan, Yun-Ruo Yang, Zhi Chen & Zhi-Xin Liao,Two new alkaloids from Tibetan medicine of Hypecoum leptocarpum,Natural Product Research,(2021)doi.org/10.1080/14786419.2021.1937154
5. Yan Feng, Israa Assani, Chun-Gu Wang, Pei-Lei Hou, Shi-Feng Zhao, Hao-Jie Ye, Rui-Chen Li, Jin-Bin Zhang, and Zhi-Xin Liao. A New Aliphatic Ketone, Chemical Composition, Antibacterial, Antioxidant and In Vitro Cytotoxic Activities of Lepidium latifolium. ChemistrySelect (2020)5: 8992-8997.
6. Israa Assani, Ying Du, Chun-Gu Wang, Lei Chen, Pei-Lei Hou, Shi-Feng Zhao, Yan Feng, Ling-Fei Liu, Bo Sun, Yan Li, Zhi-Xin Liao, and Ri-Zhen Huang. Anti-proliferative effects of diterpenoids from Sagittaria trifolia L. tubers on colon cancer cells by targeting the NF-κB pathway. Food & Function (2020)11: 7717-7726.
7. Shifeng Zhao, Yuan He, Chungu Wang, Israa Assani, Peilei Hou, Yan Feng, Juanjuan Yang, Yehua Wang, Zhi-Xin Liao, and Songdong Shen. Isolation, Characterization and Bioactive Properties of Alkali-Extracted Polysaccharides from Enteromorpha prolifera. Marine Drugs (2020)18: 552.
8. Xinzhu Wang, Liya Zhao, Chao Liu, Jun Qi, Peipei Zhao, Zhaoming Liu, Chunlei Li, Yingying Hu, Xin Yin, Xin Liu, Zhi-Xin Liao, Lixin Zhang, and Xuekui Xia. New Tetramic Acids Comprising of Decalin and Pyridones From Chaetomium olivaceum SD-80AWith Antimicrobial Activity. Frontiers in Microbiology(2020)10: 2958.
9. Ri-Zhen Huang, Gui-Bin Liang, Mei-Shan Li, Yi-Lin Fang, Shi-Feng Zhao, Mei-Mei Zhou, Zhi-Xin Liao, Jing Sun, and Heng-Shan Wang. Synthesis and discovery of asiatic acid based 1,2,3-triazole derivatives as antitumor agents blocking NF-κB activation and cell migration. Medchemomm (2019)10: 584-597.
10. Huang, RZ; Jin, L; Wang, CG; Xu, XJ; Du, Y; Liao, N; Ji, M; Liao, ZX; Wang, HS. A pentacyclic triterpene derivative possessing polyhydroxyl ring A suppresses growth of HeLa cells by reactive oxygen species-dependent NF-kappa B pathway. European Journal of Pharmacology. 2018. 838. 157-169
11. Zhang, J; Huang, RZ; Cao, HJ; Cheng, AW; Jiang, CS; Liao, ZX; Liu, C; Sun, JY. Chemical composition, in vitro anti-tumor activities and related mechanisms of the essential oil from the roots of Potentilla discolor. INDUSTRIAL CROPS AND PRODUCTS. 2018. 113. 19-27.
12. Jiang, W; Huang, RZ; Zhang, J; Guo, T; Zhang, MT; Huang, XC; Zhang, B; Liao, ZX; Sun, J; Wang, HS. Discovery of antitumor ursolic acid long-chain diamine derivatives as potent inhibitors of NF-kappa B. BIOORGANIC CHEMISTRY. 2018. 79. 265-276.
13. Huang, RZ ; Liang, GB; Huang, XC ; Zhang, B; Zhou, MM ; Liao, ZX; Wang, HS , Discovery of dehydroabietic acid sulfonamide based derivatives as selective matrix metalloproteinases inactivators that inhibit cell migration and proliferation, European Journal of Medicinal Chemistry, 2017,138, 979-992.
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